作者:Yiyun Wang;Youwei Xu;Zhonghui Zheng;Min Xue;Zihui Meng;Zhibin Xu;Jiarong Li;Qing Lin (1School of Chemistry and Chemical Engineering, Beijing Institute of Technology, Beijing 102488, China;2Shandong Xinhua Pharmaceutical Co., Ltd., Zibo 255086, China;3ReadCrystal Biotech Co., Ltd., Suzhou 215505, China)
出处:Crystals 2022
关键词:Parkinson’s disease;istradefylline;solubility;crystal form;dissolution
摘要:Istradefylline as a selective adenosine A2A-receptor antagonist is clinically used to treat Parkinson’s disease and improve dysk ...
作者:Yiyun Wang;Xiaofang Lv;Zihui Meng;Zhibin Xu;Zhonghui Zheng;Jiarong Li;Min Xue (1 School of Chemistry and Chemical Engineering, Beijing Institute of Technology, Beijing 100081, China 2 Shandong Xinhua Pharmaceutical Co., Ltd., No.1 Lutai Avenue, Zibo 255086, China Authors to whom correspondence should be addressed.)
出处:Crystals 2022
关键词:baloxavir marboxil;intermediate;synthesis;sulfonate resin solid acid;microwave irradiation
摘要:The compound (±)-12aR-12-[(11S)-7,8-difluoro-6,11-dihydrodibenzo[b,e]thiepin-11-yl]-7-hydroxy-3,4,12,12a-tetrahydro-1H-[1,4]oxazino[3,4-c]pyrid ...
作者:Lu Hong Yan,Li Jia Rong,Yang De Li (Chemical Engineering and Environment Beijing Institute of Technology,100081)
出处:中国化学快报(英文版) 2015
关键词:Cucurbituril;Nitroform;Nitrolysis;Homologues
作者:Yiyun Wang1;Jiaru Wang1;Hui Wu2;Longyao Cui2;Zihui Meng1;Zhibin Xu1;Zhonghui Zheng2;Jiarong Li1; (1School of Chemistry and Chemical Engineering, Beijing Institute of Technology, Beijing 100081, China;2Shandong Xinhua Pharmaceutical Co., Ltd., No.1Lutai Avenue, Zibo 255086, China)
出处:Crystals 2023
关键词:baloxavir;derivatives;synthesis;inhibition
摘要:Baloxavir marboxil is a creative antiviral drug for influenza A and B viruses with a novel mechanism of action. In this study, three series comprising ...
作者:Kai Zhang1 2;Yuanyuan Xu1;Shang Gao1;Jiarong Li3; (1 School of Chemical Engineering, Shijiazhuang University, Shijiazhuang, Hebei, China. 2 Shijiazhuang Key Laboratory of Target Drug Research and Pharmacodynamic Evaluation, Shijiazhuang, Hebei, China. 3 School of Chemistry and Chemical Engineering, Beijing Institute of Technology, Beijing, China.)
出处:Natural product research 2023
关键词:Spinetoram;derivatization;insecticidal activity;synthesis.
摘要:As the second generation commercial product of spinosyns, spinetoram not only has obvious insecticidal effect on vegetable crops, but also can effecti ...
作者:Na Wang1;Yaxin Guo1;Jiarong Li1;Shufeng Pang1;
出处:Atmospheric Environment 2022
关键词:Amino acid;Ammonium nitrate;ATR-FTIR;Hygroscopic properties;Microscopy technology
摘要:Water-soluble amino acids have been confirmed as effective cloud condensation nuclei (CCN) materials. While their influence on the hygroscopicity of n ...
作者:张凯1,2;,徐元媛1;,高尚1;,李加荣3; (1石家庄学院;2石家庄市靶点药物研究与药效学评价重点实验室;3北京理工大学)
出处:现代农药 2024
关键词:乙基多杀菌素;多杀霉素;研究进展
摘要:多杀菌素类化合物是一类新型高效的生物源杀虫剂,对多种害虫具有显著的活性抑制作用。多杀霉素(spinosad)和乙基多杀菌素(spinetoram)为多杀菌素类化合物第1代和第2代商业化产品,具有杀虫活性高、降解速度快、对环境友好以及对非靶标生物毒性低等特点。本文着重对乙基多杀菌素的理化性质、杀虫机制 ...
作者:李加荣,陈博仁,欧育湘,范广裕,崔秀山 (北京理工大学)
出处:北京理工大学学报 1993